产品信息
抗原名称
PDK-1
商品描述
BX-517 is a potent and selective inhibitor of PDK1 that binds to the ATP binding pocket of the protein (IC50 = 6 nM).
分子量
282.3
纯度
>98%
可溶性
DMSO: ≥ 27 mg/mL
In vitro(体外研究)
BX-517 blocks activation of Akt in tumor cells, is potent with IC50 of 0.1-1.0 μM. BX-517 blocks AKT2 activation in cells with submicromolar potency. BX-517 is 100-fold selective or better against a panel of seven additional Ser/Thr and Tyr kinases.
背景
别名
BX517, BX 517
分子式
C15H14N4O2
CAS号
850717-64-5
制备和贮存
保存方式
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
参考图片
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