产品信息
抗原名称
Cannabinoid Receptor
商品描述
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
分子量
572.51
纯度
98%
可溶性
DMSO : 250 mg/mL (436.67 mM; Need ultrasonic)
In vivo(体内研究)
JD5037 (3 mg/kg/d, i.p.) induces equal reductions in body weight, attenuates the HFD-induced hyperglycemia, and reduces the HFD-induced hepatic injury and steatosis in obese Magel2-null mice. JD5037 (3 mg/kg/day, p.o.) significantly reduces the size of tumors and abrogates the tumor in DEN-treated mice. JD5037 attenuates the AEA levels in HCC samples from mice.
背景
分子式
C27H27Cl2N5O3S
CAS号
1392116-14-1
制备和贮存
保存方式
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
参考图片
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