产品信息
商品描述
GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.
分子量
632.61
纯度
>98%
可溶性
10 mM in DMSO
背景
别名
GSK-256066, GSK 256066
分子式
C29H27F3N4O7S
CAS号
1415560-64-3
制备和贮存
保存方式
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
参考图片
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